Gold catalysis on immobilized substrates: a heteroannulation approach to the solid-supported synthesis of indoles.
نویسندگان
چکیده
A gold-catalyzed cyclization of immobilized 2-alkynylanilines was developed as the key step in the synthetic sequence for the preparation of 2-substituted indoles. These results demonstrate the potential of the unexplored combination of gold catalysis and solid-phase organic synthesis.
منابع مشابه
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عنوان ژورنال:
- Organic & biomolecular chemistry
دوره 10 13 شماره
صفحات -
تاریخ انتشار 2012